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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7147 | Valbenazine | NBI-98854 | Monoamine Transporter |
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia. | |||
T0719 | Tetrabenazine | Xenazine,Ro 1-9569 | Others , Dopamine Receptor , Monoamine Transporter |
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high... | |||
T13133 | Tetrabenazine Metabolite | (-)-β-Dihydrotetrabenazine,(-)-β-HTBZ | Monoamine Transporter |
Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine. Tetrabenazine Metabolite has a high affinity for VMAT2 with a Ki of 13.4 nM. Tetraben... | |||
T13134 | (+)-Tetrabenazine | (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ | Monoamine Transporter |
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. | |||
T25750 | Lobelane Hydrochloride | ||
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor. | |||
T79061 | VMAT2-IN-2 tosylate | Monoamine Transporter | |
VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1]. | |||
T24941 | VMAT2-IN-I HCl | VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride | |
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A. | |||
T22452 | Valbenazine tosylate | NBI-98854 | Monoamine Transporter |
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM). |