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Search Results for " vmat2 inhibitor "

8

Compounds

Cat No. Product Name Synonyms Targets
T7147 Valbenazine NBI-98854 Monoamine Transporter
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.
T0719 Tetrabenazine Xenazine,Ro 1-9569 Others , Dopamine Receptor , Monoamine Transporter
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high...
T13133 Tetrabenazine Metabolite (-)-β-Dihydrotetrabenazine,(-)-β-HTBZ Monoamine Transporter
Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine. Tetrabenazine Metabolite has a high affinity for VMAT2 with a Ki of 13.4 nM. Tetraben...
T13134 (+)-Tetrabenazine (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ Monoamine Transporter
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.
T25750 Lobelane Hydrochloride
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor.
T79061 VMAT2-IN-2 tosylate Monoamine Transporter
VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].
T24941 VMAT2-IN-I HCl VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.
T22452 Valbenazine tosylate NBI-98854 Monoamine Transporter
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).
TargetMol